SHU 9119 acetate
Product Specifications
Target
Melanocortin Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Purity
0.998
Bioactivity
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC4R and MC5R is 0.23, 0.06, and 0.09 nM respectively.
Smiles
CCCC[C@@H](C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@@H](NC([C@@H](NC([C@H](NC([C@@H](NC1=O)CC2=CNC=N2)=O)CC3=CC4=CC=CC=C4C=C3)=O)CCCNC(N)=N)=O)CC5=CNC6=C5C=CC=C6)=O)=O)=O)NC(C)=O.CC(O)=O
Molecular Formula
C56H75N15O11
Molecular Weight
1134.29
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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