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PF-06465469

Product Specifications

CAS Number

1407966-77-1

Target

CXCR|||BTK|||PD-1/PD-L1|||Tyrosine Kinases|||LAG-3

Related Pathways

Autophagy|||Cell Cycle/Checkpoint|||Immunology/Inflammation|||Tyrosine Kinase/Adaptors|||Apoptosis|||GPCR/G Protein|||Angiogenesis

Bioactivity

PF-06465469 is a covalent ITK inhibitor (IC?? = 2 nM) that also inhibits BTK. PF-06465469 suppresses CXCL12-mediated cell migration, decreases PD-1 and LAG-3 expression. PF-06465469 shows strong potential application in leukemia and T-cell lymphoma research.

Smiles

NC1=C2C(=NN(C2=NC=N1)[C@H]3CN(C(C=C)=O)CCC3)C4=CC(C(NC5=CC(C)=C(C(C)C)C=C5)=O)=CC=C4

Molecular Formula

C30H33N7O2

Molecular Weight

523.63

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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