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PF-03654746

Product Specifications

CAS Number

935840-31-6

Target

Histamine Receptor

Related Pathways

GPCR/G Protein, Immunology/Inflammation, Neuroscience

Purity

0.9957

Bioactivity

PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease. PF-03654746 can be used in studies about the treatment of allergic rhinitis.

Smiles

F[C@@]1(C[C@@H](C(NCC)=O)C1)C2=CC(F)=C(CN3CCCC3)C=C2

Molecular Formula

C18H24F2N2O

Molecular Weight

322.39

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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