PF-03654746
Product Specifications
CAS Number
935840-31-6
Target
Histamine Receptor
Related Pathways
GPCR/G Protein, Immunology/Inflammation, Neuroscience
Purity
0.9957
Bioactivity
PF-03654746 is a selective antagonist of the histamine H3 receptor. PF-03654746 improves cognitive efficacy and disease-modifying effects in Alzheimer's disease. PF-03654746 can be used in studies about the treatment of allergic rhinitis.
Smiles
F[C@@]1(C[C@@H](C(NCC)=O)C1)C2=CC(F)=C(CN3CCCC3)C=C2
Molecular Formula
C18H24F2N2O
Molecular Weight
322.39
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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