Opiranserin
Product Specifications
CAS Number
1441000-45-8
Target
GlyT, P2X Receptor, 5-HT Receptor
Related Pathways
Membrane transporter/Ion channel, GPCR/G Protein, Neuroscience
Bioactivity
Opiranserin is a development as an injectable agent for the treatment of postoperative pain. Opiranserin is a non-opioid and non-NSAID analgesic candidate and is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A) (IC50s: 0.86 and 1.3 μM, respectively) . Opiranserin displays antagonistic activity on rP2X3 (IC50=0.87 μM) .
Smiles
C(NC(=O)C1=CC(OC)=C(OCCCC)C(OC)=C1)C2(N(C)C)CCOCC2
Molecular Formula
C21H34N2O5
Molecular Weight
394.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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