OP-3633
Product Specifications
CAS Number
2102494-14-2
Target
Others, Glucocorticoid Receptor
Related Pathways
Endocrinology/Hormones, Others
Bioactivity
OP-3633 is an effective and selective steroidal glucocorticoid receptor (GR) antagonist (IC50: 29 nM) . OP-3633 shows low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism. It also has an inhibition of GR transcriptional activity.
Smiles
C[C@@]12[C@@]3([C@]([C@]4([C@](C)(C[C@@]3(C5=CC=C(N(C)C)C=C5)[H])[C@@](C#CC)(O)CC4)[H])(CCC1=CC(=O)CC2)[H])[H]
Molecular Formula
C30H39NO2
Molecular Weight
445.64
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS642529-01 0.2 mL
PI3KC3 (S34) (PIK3C3, VPS34, Phosphatidylinositol 3-kinase catalytic subunit type 3, Phosphatidylinositol 3-kinase p100 subunit, Phosphoinositide-3-kinase class 3, hVps34)
Sign In for Pricing
View Details MBS642529-02 5x 0.2 mL
PI3KC3 (S34) (PIK3C3, VPS34, Phosphatidylinositol 3-kinase catalytic subunit type 3, Phosphatidylinositol 3-kinase p100 subunit, Phosphoinositide-3-kinase class 3, hVps34)
Sign In for Pricing
View Details 
MBS9904309-01 48 Well
Monkey Zinc Finger Protein 516 (ZNF516) ELISA Kit
Sign In for Pricing
View Details MBS9904309-02 96 Well
Monkey Zinc Finger Protein 516 (ZNF516) ELISA Kit
Sign In for Pricing
View Details