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PF-02575799

Product Specifications

CAS Number

863491-70-7

Target

Adenosine Receptor, MTP, MTP

Related Pathways

Proteases/Proteasome, GPCR/G Protein, Neuroscience, Metabolism

Bioactivity

PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM) .

Smiles

C(NC1=NC2=C(C=C1)C=C(C(N[C@H](C(N(CC3=CC=C(F)C=C3)C)=O)C4=CC=CC=C4)=O)C=C2)(=O)C5=C(C=CC=C5)C6=CC=C(OC(C)C)C=C6

Molecular Formula

C42H37FN4O4

Molecular Weight

680.77

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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