PF-02575799
Product Specifications
CAS Number
863491-70-7
Target
Adenosine Receptor, MTP, MTP
Related Pathways
Proteases/Proteasome, GPCR/G Protein, Neuroscience, Metabolism
Bioactivity
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM) .
Smiles
C(NC1=NC2=C(C=C1)C=C(C(N[C@H](C(N(CC3=CC=C(F)C=C3)C)=O)C4=CC=CC=C4)=O)C=C2)(=O)C5=C(C=CC=C5)C6=CC=C(OC(C)C)C=C6
Molecular Formula
C42H37FN4O4
Molecular Weight
680.77
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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