MS417
Product Specifications
CAS Number
916489-36-6
Target
HIV Protease|||Epigenetic Reader Domain
Related Pathways
Microbiology/Virology|||Chromatin/Epigenetic|||Proteases/Proteasome
Purity
0.9988
Bioactivity
MS417 (GTPL7512) is an inhibitor of BET-specific BRD4 (BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively), with weak selectivity at CBP BRD with IC50 of 32.7 ?M.
Smiles
COC(=O)C[C@@H]1N=C(c2c(C)c(C)sc2-n2c(C)nnc12)c1ccc(Cl)cc1
Molecular Formula
C20H19ClN4O2S
Molecular Weight
414.91
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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