MRS 1754
Product Specifications
CAS Number
264622-58-4
Target
Adenosine Receptor
Related Pathways
Neuroscience|||GPCR/G Protein
Purity
0.993
Bioactivity
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor, exhibiting very low affinity for A1 and A3 receptors in both humans and rats.
Smiles
CCCn1c2[nH]c(nc2c(=O)n(CCC)c1=O)-c1ccc(OCC(=O)Nc2ccc(cc2)C#N)cc1
Molecular Formula
C26H26N6O4
Molecular Weight
486.52
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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