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MRS-1191

Product Specifications

CAS Number

185222-90-6

Target

Others, Adenosine Receptor

Related Pathways

Others, Neuroscience, GPCR/G Protein

Bioactivity

MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells) .

Smiles

CCOC(=O)C1=C(C)NC(=C(C1C#Cc1ccccc1)C(=O)OCc1ccccc1)c1ccccc1

Molecular Formula

C31H27NO4

Molecular Weight

477.55

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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