LP-935509
Product Specifications
CAS Number
1454555-29-3
Target
AAK1, AAK1 (AP2 associated kinase 1), Serine/threonin kinase, SARS-CoV
Related Pathways
Microbiology/Virology, Metabolism, Cell Cycle/Checkpoint, Neuroscience
Purity
0.9964
Bioactivity
LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1) with an IC50 of 3.3 nM and a Ki of 0.9 nM. LP-935509 is a potent inhibitor of BIKE (IC50 of 14 nM) and a moderate inhibitor of GAK (IC50 of 320±40 nM) .
Smiles
COc1ncccc1-c1cnn2ccc(nc12)N1CCN(CC1)C(=O)OC(C)C
Molecular Formula
C20H24N6O3
Molecular Weight
396.44
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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