Linopirdine
Product Specifications
CAS Number
105431-72-9
Target
Potassium Channel, TRP/TRPV Channel
Related Pathways
Membrane transporter/Ion channel
Purity
0.9992
Bioactivity
Linopirdine (DuP 996) is a TRPV1 agonist. Linopirdine is an orally active and selective M-type K+ current (IM; Kv7; KCNQ Channels) inhibitor (IC50: 2.4 μM) . Linopirdine is a cognitive enhancer. It acts by stimulating release of acetylcholine and other neurotransmitters.Linopirdine is a putative cognition-enhancing drug that increases acetylcholine release in rat brain tissue.
Smiles
O=C1N(c2ccccc2C1(Cc1ccncc1)Cc1ccncc1)c1ccccc1
Molecular Formula
C26H21N3O
Molecular Weight
391.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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