Larotaxel

Product Specifications

CAS Number

156294-36-9

Target

P-gp|||Apoptosis

Related Pathways

Apoptosis|||Membrane transporter/Ion channel|||Neuroscience

Purity

0.9922

Bioactivity

Larotaxel (XRP9881) is a taxane analogue with anticancer activity that promotes tubulin assembly and stabilizes microtubules, inducing apoptosis. It crosses the blood-brain barrier and has a higher affinity for Docetaxel than P-glycoprotein 1, making it useful for studying breast and bladder cancer.

Smiles

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