KDM5A-IN-1
Product Specifications
CAS Number
1905481-36-8
Target
Histone Demethylase
Related Pathways
Chromatin/Epigenetic
Purity
>99.99%
Bioactivity
KDM5A-IN-1 is an orally available, potent and selective inhibitor of the pan-histidine lysine demethylase 5 KDM5, inhibiting KDM5A, KDM5B, and KDM5C with IC50 values of 45 nM, 56 nM, and 55 nM, respectively.KDM5A-IN-1 inhibits PC9 H3K4Me3, and may be useful in cancer research.
Smiles
CC(C)c1cc([nH]n1)C(=O)N1CC[C@H](C1)NC(=O)C1CC1
Molecular Formula
C15H22N4O2
Molecular Weight
290.36
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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