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JTE-013

Product Specifications

CAS Number

383150-41-2

Target

LPL Receptor, Apoptosis, S1P Receptor

Related Pathways

Apoptosis, GPCR/G Protein

Purity

0.9965

Bioactivity

JTE-013 is an effective and specific antagonist of S1P2. JTE-013 suppresses the specific binding of radiolabeled S1P to human and rat S1P2 (IC50s: 17 nM and 22 nM, respectively) .

Smiles

CC(C)c1cc(NNC(=O)Nc2cc(Cl)nc(Cl)c2)nc2n(C)nc(C)c12

Molecular Formula

C17H19Cl2N7O

Molecular Weight

408.29

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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