GS-626510
Product Specifications
CAS Number
1637770-13-8
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Bioactivity
GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2) .
Smiles
Cc1noc(C)c1-c1cc(-c2c(C)ccc3ncccc23)c2[nH]c(nc2c1)C1CC1
Molecular Formula
C25H22N4O
Molecular Weight
394.47
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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