GNE-781
Product Specifications
CAS Number
1936422-33-1
Target
Epigenetic Reader Domain, Histone Acetyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9992
Bioactivity
GNE-781 is a highly potent and selective inhibitor of CBP (IC50: 0.94 nM in TR-FRET assay) . GNE-781 also inhibits BRET and BRD4 (1) (IC50s: 6.2 nM and 5100 nM, respectively) .
Smiles
CNC(=O)N1CCc2c(C1)c(nn2C1CCOCC1)N1CCCc2cc(-c3cnn(C)c3)c(cc12)C(F)F
Molecular Formula
C27H33F2N7O2
Molecular Weight
525.59
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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