What is the catalog number for GNE-049?

The catalog number for GNE-049 is T15397.

What sizes are available for GNE-049?

GNE-049 is available in the following size(s): 1 mg, 5 mg, 1 mL - 10 mM (in DMSO), 10 mg, 25 mg, 50 mg.

How many pack sizes does GNE-049 come in?

GNE-049 is available in 6 different pack sizes.

GNE-049 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GNE-049?

GNE-049 is manufactured by Molfinity.

What is the estimated delivery time for GNE-049?

Estimated delivery time for GNE-049 is approximately 10 business day(s), depending on your location.

GNE-049

Product Specifications

CAS Number

1936421-41-8

Target

Epigenetic Reader Domain, Histone Acetyltransferase

Related Pathways

Chromatin/Epigenetic

Purity

0.9867

Bioactivity

GNE-049 is a highly selective and potent inhibitor designed to target the CREB-binding protein (CBP) with high affinity, exhibiting an IC50 of 1.1 nM for the suppression of BRET and BRD4 activity, which consequently blocks prostate cancer cell proliferation in both in vitro and in vivo models.