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GLP-1R Antagonist 1

Product Specifications

CAS Number

488097-06-9

Target

Glucagon Receptor

Related Pathways

GPCR/G Protein

Purity

0.9984

Bioactivity

GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM) .

Smiles

Cn1c2NC(=NC(c2c(=O)n(C)c1=O)(C(F)(F)F)C(F)(F)F)c1ccc(Cl)cc1

Molecular Formula

C16H11ClF6N4O2

Molecular Weight

440.73

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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