GLP-1R Antagonist 1
Product Specifications
CAS Number
488097-06-9
Target
Glucagon Receptor
Related Pathways
GPCR/G Protein
Purity
0.9984
Bioactivity
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM) .
Smiles
Cn1c2NC(=NC(c2c(=O)n(C)c1=O)(C(F)(F)F)C(F)(F)F)c1ccc(Cl)cc1
Molecular Formula
C16H11ClF6N4O2
Molecular Weight
440.73
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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