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MAK683

Product Specifications

CAS Number

1951408-58-4

Target

Histone Methyltransferase

Related Pathways

Chromatin/Epigenetic

Purity

0.9992

Bioactivity

MAK683 is an inhibitor of embryonic ectoderm development (EED) (IC50s: 59, 89, 26 nM in EED Alphascreen binding, LC-MS and ELISA assay) .

Smiles

Cc1ncccc1-c1cnc(NCc2c3CCOc3ccc2F)n2cnnc12

Molecular Formula

C20H17FN6O

Molecular Weight

376.39

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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