CCG-63808
Product Specifications
CAS Number
620113-73-7
Target
GTPase
Related Pathways
GPCR/G Protein
Purity
0.9
Bioactivity
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins, dose-dependently inhibiting the TR-FRET signal between RGS4-AF488 and Tb-Gαo with an IC50 value of 1.9 μM.
Smiles
Cc1cccn2c1nc(Oc1ccc(F)cc1)c(\C=C(/C#N)c1nc3ccccc3s1)c2=O
Molecular Formula
C25H15FN4O2S
Molecular Weight
454.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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