CCG-63808

Product Specifications

CAS Number

620113-73-7

Target

GTPase

Related Pathways

GPCR/G Protein

Purity

0.9

Bioactivity

CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins, dose-dependently inhibiting the TR-FRET signal between RGS4-AF488 and Tb-Gαo with an IC50 value of 1.9 μM.

Smiles

Cc1cccn2c1nc(Oc1ccc(F)cc1)c(\C=C(/C#N)c1nc3ccccc3s1)c2=O

Molecular Formula

C25H15FN4O2S

Molecular Weight

454.48

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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