BTRX-335140
Product Specifications
CAS Number
2244614-14-8
Target
Opioid Receptor
Related Pathways
GPCR/G Protein, Endocrinology/Hormones, Neuroscience
Purity
0.9989
Bioactivity
BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity against κOR, μOR, and δOR with IC50 values of 0.8, 110, and 6500 nM, respectively.
Smiles
CCc1cc(F)c2nc(N3CCC(CC3)NC3CCOCC3)c(-c3nc(C)no3)c(C)c2c1
Molecular Formula
C25H32FN5O2
Molecular Weight
453.55
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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