BMS-986158
Product Specifications
CAS Number
1800340-40-2
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9878
Bioactivity
BMS-986158 is a highly effective BET inhibitor, demonstrating IC50 values of 6.6 nM in NCI-H211 small cell lung cancer (SCLC) cells and 5 nM in MDA-MB231 triple negative breast cancer (TNBC) cells.
Smiles
Cc1nnn(C)c1-c1cnc2c(c1)n([C@@H](C1CCOCC1)c1ccccc1)c1cc(ccc21)C(C)(C)O
Molecular Formula
C30H33N5O2
Molecular Weight
495.62
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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