BMS-819881

Product Specifications

CAS Number

1197420-05-5

Target

Cytochromes P450|||Melanin-concentrating Hormone Receptor (MCHR) |||GPCR

Related Pathways

GPCR/G Protein|||Endocrinology/Hormones|||Metabolism

Bioactivity

BMS-819881, a melanin-concentrating hormone receptor 1 (MCHR1) antagonist, binds rat MCHR1 with a Ki of 7 nM, and is selective and potent for CYP3A4 activity with an EC50 of 13 ?M.

Smiles

O=C1C2=C(C=C(S2)C3=CC=C(Cl)C=C3)N=CN1C4=CC(OC)=C(OC[C@H](O)C5CC5)C=C4

Molecular Formula

C24H21ClN2O4S

Molecular Weight

468.95

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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