AZD1979
Product Specifications
CAS Number
1254035-84-1
Target
GPCR, Melanin-concentrating Hormone Receptor (MCHR)
Related Pathways
GPCR/G Protein, Endocrinology/Hormones
Purity
0.9972
Bioactivity
AZD1979 is a highly potent MCHR1 (Melanin-concentrating hormone receptor 1) antagonist with an IC50 of 12 nM, exhibiting improved central nervous system (CNS) exposure and enhanced insulin sensitivity in steady-state model assessments, making it suitable for the treatment of obesity.
Smiles
O=C(C1=NN=C(O1)C=2C=CC(OC)=CC2)N3CC(OC4=CC=C(C=C4)CN5CC6(COC6)C5)C3
Molecular Formula
C25H26N4O5
Molecular Weight
462.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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