Autotaxin-IN-1
Product Specifications
CAS Number
1619971-30-0
Target
PDE
Related Pathways
Metabolism
Bioactivity
Autotaxin-IN-1 is a potent autotaxin inhibitor used in the treatment of osteoarthritis pain. It exhibits favorable potency (IC50=2.2 nM), pharmacokinetic (PK) properties, and a robust PK/pharmacodynamic (PD) relationship[1].
Smiles
C(COCCC1=CN=NN1)(=O)N2CC=3C(C2)=CN=C(NC4CC=5C(C4)=CC=CC5)N3
Molecular Formula
C21H23N7O2
Molecular Weight
405.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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