ARP-100
Product Specifications
CAS Number
704888-90-4
Target
MMP
Related Pathways
Proteases/Proteasome
Purity
0.9834
Bioactivity
ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM) . ARP-100 interacts with the S1' pocket of MMP-2 and exhibits anti-invasive properties in an in vitro invasion Matrigel model. ARP-100 has low inhibitory activity against MMP-1 (>50 μM), MMP-3 (4.5 μM), MMP-7 (>50 μM) and MMP-9 (0.2 μM) [1][2].
Smiles
CC(C)ON(CC(=O)NO)S(=O)(=O)c1ccc(cc1)-c1ccccc1
Molecular Formula
C17H20N2O5S
Molecular Weight
364.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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