ARP-100
Product Specifications
CAS Number
704888-90-4
Target
MMP
Related Pathways
Proteases/Proteasome
Purity
0.9834
Bioactivity
ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM) . ARP-100 interacts with the S1' pocket of MMP-2 and exhibits anti-invasive properties in an in vitro invasion Matrigel model. ARP-100 has low inhibitory activity against MMP-1 (>50 μM), MMP-3 (4.5 μM), MMP-7 (>50 μM) and MMP-9 (0.2 μM) [1][2].
Smiles
CC(C)ON(CC(=O)NO)S(=O)(=O)c1ccc(cc1)-c1ccccc1
Molecular Formula
C17H20N2O5S
Molecular Weight
364.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS1374069 Inquire
Recombinant Salmonella typhimurium Chaperone protein hscA (hscA), partial
Sign In for Pricing
View Details 
GTR10449527 96 Well
Guinea Pig Early Growth Response Protein 3 ELISA kit
Sign In for Pricing
View Details 
RC201743L4 10 µg
IKK gamma (IKBKG) (NM_003639) Human Tagged Lenti ORF Clone
Sign In for Pricing
View Details 