1G244
Product Specifications
CAS Number
847928-32-9
Target
Apoptosis, Proteasome
Related Pathways
Ubiquitination, Proteases/Proteasome, Apoptosis
Purity
0.9914
Bioactivity
1G244 is an inhibitor of DPP8/9 with antiatherosclerotic and antimyeloma properties. 1G244 had the IC50 values of 14 and 53 nM against DPP8 and DPP9, and The Ki values for 1G244 were 0.9 and 4.2 nM for DPP8 and DPP9
Smiles
N[C@@H](CC(=O)N1CCN(CC1)C(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)N1Cc2ccccc2C1
Molecular Formula
C29H30F2N4O2
Molecular Weight
504.57
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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