MS1943
Product Specifications
CAS Number
2225938-17-8
Target
PROTACs, Histone Methyltransferase, Apoptosis
Related Pathways
Chromatin/Epigenetic, PROTAC, Apoptosis
Purity
0.9826
Bioactivity
MS1943 is a orally bioavailable EZH2 selective degrader (IC50 of 120 nM) .
Smiles
CC(C)n1ncc2c(cc(cc12)-c1ccc(nc1)N1CCN(CCNC(=O)CC23CC4CC(CC(C4)C2)C3)CC1)C(=O)NCc1c(C)cc(C)[nH]c1=O
Molecular Formula
C42H54N8O3
Molecular Weight
718.93
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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