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CCG258208

Product Specifications

CAS Number

2055990-90-2

Target

GRK

Related Pathways

GPCR/G Protein

Bioactivity

GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM) .

Smiles

C(OC=1C=C2C(=CC1)OCO2)[C@H]3[C@@H](CCNC3)C4=CC(C(NCC=5C=CNN5)=O)=C(F)C=C4

Molecular Formula

C24H25FN4O4

Molecular Weight

452.48

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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