CCG258208
Product Specifications
CAS Number
2055990-90-2
Target
GRK
Related Pathways
GPCR/G Protein
Bioactivity
GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM) .
Smiles
C(OC=1C=C2C(=CC1)OCO2)[C@H]3[C@@H](CCNC3)C4=CC(C(NCC=5C=CNN5)=O)=C(F)C=C4
Molecular Formula
C24H25FN4O4
Molecular Weight
452.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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