ZEN-3862
Product Specifications
CAS Number
1952264-33-3
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.971
Bioactivity
ZEN-3862 (Willardiine) is an inhibitor of BET (IC50s of 0.16 and 0.13 μM for BRD4 (BD1) and BRD4 (BD2), respectively) . ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.
Smiles
CC=1C(C2=CN(CC3=CC(F)=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1
Molecular Formula
C19H17FN2O3
Molecular Weight
340.35
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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