ZEN-3219
Product Specifications
CAS Number
1952264-34-4
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9986
Bioactivity
ZEN-3219 is a BET inhibitor, which has inhibitory effect on BRD4 (BD1), BRD4 (BD2) and BRD4 (BD1BD2) . ZEN-3219 has inhibitory effect on BRD4 (BD1), The IC50 values of BRD4 (BD2) and BRD4 (BD1BD2) were 0.48, 0.16 and 0.47 ?M, respectively. ZEN-3219 is a component of PROTAC molecule and can induce BRD4 degradation.
Smiles
CC=1C(C2=CN(CC3=CC=C(C=C3)C4CO4)C(=O)C=C2)=C(C)ON1
Molecular Formula
C19H18N2O3
Molecular Weight
322.36
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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