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Trilaciclib hydrochloride

Product Specifications

CAS Number

1977495-97-8

Target

CDK

Related Pathways

Cell Cycle/Checkpoint

Purity

0.9989

Bioactivity

Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6) .

Smiles

Cl.Cl.CN1CCN(CC1)c1ccc(Nc2ncc3cc4C(=O)NCC5(CCCCC5)n4c3n2)nc1

Molecular Formula

C24H32Cl2N8O

Molecular Weight

519.47

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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