Tenalisib
Product Specifications
CAS Number
1639417-53-0
Target
PI3K
Related Pathways
PI3K/Akt/mTOR signaling
Purity
0.9971
Bioactivity
Tenalisib (RP6530) (RP6530) is a potent and selective inhibitor of PI3Kδ and PI3Kγ (IC50 values of 25 and 33 nM, respectively.)
Smiles
CC[C@H](Nc1ncnc2nc[nH]c12)c1oc2ccccc2c(=O)c1-c1cccc(F)c1
Molecular Formula
C23H18FN5O2
Molecular Weight
415.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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