SJB3-019A
Product Specifications
CAS Number
2070015-29-9
Target
DUB
Related Pathways
DNA Damage/DNA Repair, Cell Cycle/Checkpoint, Ubiquitination
Purity
0.9975
Bioactivity
SJB3-019A is a potent, potent and novel ubiquitin-specific protease 1 (USP1) inhibitor, which promotes ID1 degradation and cytotoxicity in K562 cells 5 times more than SJB2-043, with IC50 of 0.0781 μM. SJB3-019A inhibits cell proliferation and causes cell apoptosis.
Smiles
O=C1c2nc(oc2C(=O)c2ccccc12)-c1cccnc1
Molecular Formula
C16H8N2O3
Molecular Weight
276.25
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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