Amcenestrant
Product Specifications
CAS Number
2114339-57-8
Target
Estrogen/progestogen Receptor, Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Purity
0.99
Bioactivity
Amcenestrant (SAR439859) is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD) . SAR439859 is a potent antagonist of ER (with an EC50 of 0.2 nM for ERα degradation) .
Smiles
OC(=O)c1ccc2c(CCCC(c3ccc(Cl)cc3Cl)=C2c2ccc(O[C@H]3CCN(CCCF)C3)cc2)c1
Molecular Formula
C31H30Cl2FNO3
Molecular Weight
554.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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