RORγt Inverse agonist 3
Product Specifications
CAS Number
2364429-77-4
Target
Others, ROR
Related Pathways
Others, Metabolism
Bioactivity
RORγt Inverse Agonist 3 is a potent, selective, and orally active inverse agonist of RORγ with EC50 values of 0.22 μM for hRORγ and 0.15 μM for RORγt (human IL-17 cells), respectively.
Smiles
CNC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc(Cl)c(COc2cccc3c(cc(nc23)C(C)C)-c2cncn2C)c1Cl
Molecular Formula
C29H31Cl2N5O4S
Molecular Weight
616.56
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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