(Rac) -VU 6008667
Product Specifications
CAS Number
2092917-63-8
Target
AChR
Related Pathways
Neuroscience
Purity
0.9982
Bioactivity
(Rac) -VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.
Smiles
C(=O)(N1C2(C=3C(C(=O)N2CC1)=CC=CC3)C4=CC(C)=C(Cl)C=C4)C5=CC(F)=C(F)C=C5
Molecular Formula
C24H17ClF2N2O2
Molecular Weight
438.85
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS1396427-01 0.02 mg (E-Coli)
Recombinant Corynebacterium jeikeium Phosphoglycerate kinase (pgk)
Sign In for Pricing
View Details MBS1396427-02 0.02 mg (Yeast)
Recombinant Corynebacterium jeikeium Phosphoglycerate kinase (pgk)
Sign In for Pricing
View Details MBS1396427-03 0.1 mg (E-Coli)
Recombinant Corynebacterium jeikeium Phosphoglycerate kinase (pgk)
Sign In for Pricing
View Details MBS1396427-04 0.1 mg (Yeast)
Recombinant Corynebacterium jeikeium Phosphoglycerate kinase (pgk)
Sign In for Pricing
View Details MBS1396427-05 0.02 mg (Baculovirus)
Recombinant Corynebacterium jeikeium Phosphoglycerate kinase (pgk)
Sign In for Pricing
View Details MBS1396427-06 0.02 mg (Mammalian-Cell)
Recombinant Corynebacterium jeikeium Phosphoglycerate kinase (pgk)
Sign In for Pricing
View Details