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PI3Kα/mTOR-IN-1

Product Specifications

CAS Number

1013098-90-2

Target

PI3K, mTOR

Related Pathways

PI3K/Akt/mTOR signaling

Purity

0.9989

Bioactivity

PI3Kα/mTOR-IN-1 is a potent dual inhibitor of PI3Kα/mTOR, with an IC50 of 7 nM for PI3Kα in a cell assay and Kis of 12.5 nM and 10.6 nM for mTOR and PI3Kα [in a cell-free assay], respectively.

Smiles

O=C1N(C=2C(C=C1C=3C=NNC3)=C(C)N=C(N)N2)C4CCCC4

Molecular Formula

C16H18N6O

Molecular Weight

310.35

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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