Rilzabrutinib
Product Specifications
CAS Number
1575596-29-0
Target
EGFR, HER, BTK
Related Pathways
Angiogenesis, JAK/STAT signaling, Tyrosine Kinase/Adaptors
Purity
0.9976
Bioactivity
Rilzabrutinib (PRN1008) is a reversible covalent, selective, and orally active inhibitor of Bruton's Tyrosine Kinase (BTK) with an IC50 of 1.3 nM.
Smiles
CC(C)(\C=C(/C#N)C(=O)N1CCC[C@H](C1)n1nc(-c2ccc(Oc3ccccc3)cc2F)c2c(N)ncnc12)N1CCN(CC1)C1COC1
Molecular Formula
C36H40FN9O3
Molecular Weight
665.76
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
bs-5870R-BF647 100 µL
KLK6 Polyclonal Antibody, AbBy Fluor™ 647 Conjugated
Sign In for Pricing
View Details 
K4291808 1.0 µg DNA
Dok7 sgRNA CRISPR/Cas9 All-in-One Lentivector (Mouse) (Target 3)
Sign In for Pricing
View Details 
TL311425 1 Kit
MRG15 (MORF4L1) Human shRNA Plasmid Kit (Locus ID 10933)
Sign In for Pricing
View Details