PIM1-IN-1
Product Specifications
CAS Number
1417630-95-5
Target
Pim
Related Pathways
Chromatin/Epigenetic|||JAK/STAT signaling
Bioactivity
PIM1-IN-1 is a potent and highly selective inhibitor of PIM1/3 (IC50s: 7 nM for PIM1, 5530 nM for PIM2, and 70 nM for PIM3) with antiproliferative and anti-cancer activity.
Smiles
COCCN1CCOc2c1cnn1c(nnc21)-c1ccc2cccc(NCC3CCNCC3)c2n1
Molecular Formula
C25H30N8O2
Molecular Weight
474.56
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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