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PF-04957325

Product Specifications

CAS Number

1305115-80-3

Target

PDE

Related Pathways

Metabolism

Purity

0.9902

Bioactivity

PF-04957325 is a potent and selective inhibitor of PDE8.PF-04957325 has an IC50 of 0.7 nM for PDE8A and 0.3 nM for PDE8B.PF-04957325 can be used to study autoimmune encephalomyelitis.

Smiles

Nc1nc(nc2n(C[C@H]3CN(Cc4nccs4)CCO3)nnc12)C(F)(F)F

Molecular Formula

C14H15F3N8OS

Molecular Weight

400.38

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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