PARP14 inhibitor H10
Product Specifications
CAS Number
2084811-68-5
Target
PARP|||Apoptosis
Related Pathways
Apoptosis|||Chromatin/Epigenetic|||DNA Damage/DNA Repair
Bioactivity
PARP14 inhibitor H10 is a selective inhibitor against PARP14 with IC50 of 490 nM
Smiles
NC(=O)c1cccc(NC(=O)CCC(=O)NCCc2cn(CCNS(=O)(=O)c3cccc(c3)C(O)=O)nn2)c1
Molecular Formula
C24H27N7O7S
Molecular Weight
557.58
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Curated Selection
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