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PARP14 inhibitor H10

Product Specifications

CAS Number

2084811-68-5

Target

PARP|||Apoptosis

Related Pathways

Apoptosis|||Chromatin/Epigenetic|||DNA Damage/DNA Repair

Bioactivity

PARP14 inhibitor H10 is a selective inhibitor against PARP14 with IC50 of 490 nM

Smiles

NC(=O)c1cccc(NC(=O)CCC(=O)NCCc2cn(CCNS(=O)(=O)c3cccc(c3)C(O)=O)nn2)c1

Molecular Formula

C24H27N7O7S

Molecular Weight

557.58

Shipping Conditions

Cool pack

Storage Temperature

-20°C

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