Benzquinamide
Product Specifications
CAS Number
63-12-7
Target
Adrenergic Receptor
Related Pathways
Neuroscience, GPCR/G Protein
Purity
0.9486
Bioactivity
Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer drugs in multidrug-resistant cells.The Ki values of Benzquinamide for α2A, α2B, and α2C adrenergic receptor (α2-AR) were 1,365, 691, and 545 nM, respectively. 545 nM, respectively.
Smiles
CCN(CC)C(=O)C1CN2CCc3cc(OC)c(OC)cc3C2CC1OC(C)=O
Molecular Formula
C22H32N2O5
Molecular Weight
404.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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