MK-0249
Product Specifications
CAS Number
862309-06-6
Target
Histamine Receptor
Related Pathways
Immunology/Inflammation, GPCR/G Protein, Neuroscience
Purity
0.999
Bioactivity
MK-0249 is an orally active, selective and potent histamine H3 receptor antagonist (IC50: 1.7 nM) for the study of attention-deficit and hyperactivity disorders.
Smiles
Cc1nc2cccc(c2c(=O)n1-c1ccc(OCCCN2CCCC2)cc1)C(F)(F)F
Molecular Formula
C23H24F3N3O2
Molecular Weight
431.45
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog